RGS14 prevents morphine from internalizing Mu-opioid receptors in periaqueductal gray neurons. [electronic resource]
- Cellular signalling Dec 2007
- 2558-71 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0898-6568
10.1016/j.cellsig.2007.08.003 doi
Amino Acid Sequence Analgesics, Opioid--administration & dosage Animals Calcium-Calmodulin-Dependent Protein Kinase Type 2--metabolism Disease Models, Animal Dose-Response Relationship, Drug Drug Tolerance Endocytosis--drug effects Enkephalin, Ala(2)-MePhe(4)-Gly(5)---pharmacology Enzyme Activation G-Protein-Coupled Receptor Kinases--metabolism Gene Silencing Hot Temperature--adverse effects Injections, Intraventricular Male Mice Molecular Sequence Data Morphine--administration & dosage Neurons--drug effects Oligonucleotides, Antisense--metabolism Pain--etiology Pain Measurement Pain Threshold--drug effects Periaqueductal Gray--cytology Phosphorylation RGS Proteins--genetics Receptors, Opioid, mu--agonists Serine--metabolism Synaptosomes--drug effects Time Factors