Roecker, Anthony J

Kinesin spindle protein (KSP) inhibitors. Part 8: Design and synthesis of 1,4-diaryl-4,5-dihydropyrazoles as potent inhibitors of the mitotic kinesin KSP. [electronic resource] - Bioorganic & medicinal chemistry letters Oct 2007 - 5677-82 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2007.07.074 doi


Binding Sites
Crystallography, X-Ray
Drug Design
Humans
Hydrogen--chemistry
Kinesins--antagonists & inhibitors
Mitosis--drug effects
Models, Molecular
Molecular Structure
Pyrazoles--chemical synthesis
Structure-Activity Relationship