Dual serotonin transporter inhibitor/histamine H3 antagonists: development of rigidified H3 pharmacophores. [electronic resource]
- Bioorganic & medicinal chemistry letters Oct 2007
- 5325-9 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2007.08.017 doi
5-Hydroxytryptophan--pharmacology Animals Brain--metabolism Drug Design Histamine Antagonists--chemical synthesis Humans Indicators and Reagents Rats Receptors, Histamine H3--drug effects Serotonin Antagonists--chemical synthesis Serotonin Plasma Membrane Transport Proteins--drug effects Structure-Activity Relationship Tetrahydroisoquinolines--chemical synthesis