Keith, John M

Pyrrolidino-tetrahydroisoquinolines bearing pendant heterocycles as potent dual H3 antagonist and serotonin transporter inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2007 - 4374-7 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2007.03.043 doi


Animals
Blood-Brain Barrier
Histamine H1 Antagonists--chemistry
Mice
Pyrrolidines--chemistry
Receptors, Histamine H3--drug effects
Serotonin Plasma Membrane Transport Proteins--drug effects
Structure-Activity Relationship
Tetrahydroisoquinolines--chemistry