Gurney, H

Imatinib disposition and ABCB1 (MDR1, P-glycoprotein) genotype. [electronic resource] - Clinical pharmacology and therapeutics Jul 2007 - 33-40 p. digital

Publication Type: Clinical Trial; Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

0009-9236

10.1038/sj.clpt.6100201 doi


ATP Binding Cassette Transporter, Subfamily B
ATP Binding Cassette Transporter, Subfamily B, Member 1
Adult
Aged
Aged, 80 and over
Antineoplastic Agents--administration & dosage
Benzamides
Cohort Studies
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme System--genetics
Drug Monitoring
Female
Gastrointestinal Stromal Tumors--drug therapy
Genotype
Humans
Imatinib Mesylate
Leukemia, Myelogenous, Chronic, BCR-ABL Positive--drug therapy
Male
Metabolic Clearance Rate
Middle Aged
Organic Anion Transporters--antagonists & inhibitors
Phenotype
Piperazines--administration & dosage
Polymorphism, Single Nucleotide
Protein Kinase Inhibitors--administration & dosage
Pyrimidines--administration & dosage