Gurney, H
Imatinib disposition and ABCB1 (MDR1, P-glycoprotein) genotype. [electronic resource]
- Clinical pharmacology and therapeutics Jul 2007
- 33-40 p. digital
Publication Type: Clinical Trial; Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
ISSN: 0009-9236
Standard No.: 10.1038/sj.clpt.6100201 doi
Subjects--Topical Terms: ATP Binding Cassette Transporter, Subfamily B ATP Binding Cassette Transporter, Subfamily B, Member 1 Adult Aged Aged, 80 and over Antineoplastic Agents--administration & dosage Benzamides Cohort Studies Cytochrome P-450 CYP3A Cytochrome P-450 Enzyme System--genetics Drug Monitoring Female Gastrointestinal Stromal Tumors--drug therapy Genotype Humans Imatinib Mesylate Leukemia, Myelogenous, Chronic, BCR-ABL Positive--drug therapy Male Metabolic Clearance Rate Middle Aged Organic Anion Transporters--antagonists & inhibitors Phenotype Piperazines--administration & dosage Polymorphism, Single Nucleotide Protein Kinase Inhibitors--administration & dosage Pyrimidines--administration & dosage