Yang, Jing

AZD1152, a novel and selective aurora B kinase inhibitor, induces growth arrest, apoptosis, and sensitization for tubulin depolymerizing agent or topoisomerase II inhibitor in human acute leukemia cells in vitro and in vivo. [electronic resource] - Blood Sep 2007 - 2034-40 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

0006-4971

10.1182/blood-2007-02-073700 doi


Animals
Antibiotics, Antineoplastic--pharmacology
Apoptosis--drug effects
Aurora Kinase A
Aurora Kinase B
Aurora Kinases
Case-Control Studies
Cell Cycle--drug effects
Cell Proliferation--drug effects
Colony-Forming Units Assay
Daunorubicin--pharmacology
Drug Synergism
Drug Therapy, Combination
Drug Tolerance
Enzyme Inhibitors--pharmacology
Female
Flow Cytometry
Humans
Immunoblotting
Leukemia--drug therapy
Mice
Mice, Inbred BALB C
Organophosphates--pharmacology
Protein Serine-Threonine Kinases--antagonists & inhibitors
Quinazolines--pharmacology
Thymidine--metabolism
Transplantation, Heterologous
Tubulin Modulators--pharmacology
Vincristine--pharmacology