A fragment-based approach for the discovery of isoform-specific p38alpha inhibitors. [electronic resource]
- ACS chemical biology May 2007
- 329-36 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1554-8937
10.1021/cb700025j doi
Cell Line Drug Design Humans Isoenzymes Ligands Lipopolysaccharides--pharmacology Mitogen-Activated Protein Kinase 14--antagonists & inhibitors Models, Chemical Piperidines--chemical synthesis Protein Binding Protein Kinase Inhibitors--chemical synthesis Structure-Activity Relationship Tumor Necrosis Factor-alpha--antagonists & inhibitors