Ward, P

Potent and highly selective neurokinin antagonists. [electronic resource] - Journal of medicinal chemistry Jul 1990 - 1848-51 p. digital

Publication Type: Comparative Study; Journal Article

0022-2623

10.1021/jm00169a003 doi


Amino Acid Sequence
Animals
Guinea Pigs
In Vitro Techniques
Intestinal Mucosa--metabolism
Intestines--drug effects
Molecular Sequence Data
Molecular Structure
Muscle Contraction--drug effects
Muscle, Smooth--drug effects
Neurokinin A--analogs & derivatives
Neurokinin B--analogs & derivatives
Protein Conformation
Rats
Receptors, Neurokinin-1
Receptors, Neurokinin-2
Receptors, Neurokinin-3
Receptors, Neurotransmitter--drug effects
Structure-Activity Relationship
Substance P--analogs & derivatives