In vitro and in vivo binding of neuroactive steroids to the sigma-1 receptor as measured with the positron emission tomography radioligand [18F]FPS. [electronic resource]
- Synapse (New York, N.Y.) Jul 2007
- 540-6 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
0887-4476
10.1002/syn.20369 doi
Animals Autoradiography--methods Binding, Competitive--drug effects Brain--ultrastructure Cell Membrane--diagnostic imaging Dose-Response Relationship, Drug Fluorine Radioisotopes--pharmacokinetics In Vitro Techniques Positron-Emission Tomography Protein Binding--drug effects Rats Receptors, sigma--metabolism Steroids--pharmacology Time Factors Tissue Distribution--drug effects Sigma-1 Receptor