McNally, Virginia A

Design, synthesis and enzymatic evaluation of 6-bridged imidazolyluracil derivatives as inhibitors of human thymidine phosphorylase. [electronic resource] - The Journal of pharmacy and pharmacology Apr 2007 - 537-47 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-3573

10.1211/jpp.59.4.0008 doi


Binding Sites
Drug Design
Enzyme Inhibitors--chemical synthesis
Humans
Inhibitory Concentration 50
Models, Molecular
Structure-Activity Relationship
Thymidine Phosphorylase--antagonists & inhibitors
Uracil--analogs & derivatives