Lim, Yun-Ping

Pregnane X receptor polymorphism affects CYP3A4 induction via a ligand-dependent interaction with steroid receptor coactivator-1. [electronic resource] - Pharmacogenetics and genomics May 2007 - 369-82 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1744-6872

10.1097/FPC.0b013e32803e40d7 doi


Antineoplastic Agents, Phytogenic--pharmacology
Cell Line, Tumor
Chromatography, Affinity
Clotrimazole--pharmacology
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme System--metabolism
Electrophoretic Mobility Shift Assay
Enzyme Inhibitors--pharmacology
Growth Inhibitors--pharmacology
Histone Acetyltransferases--metabolism
Humans
Immunoprecipitation
Ligands
Mutagenesis, Site-Directed
Mutation--genetics
Nuclear Receptor Coactivator 1
Paclitaxel--pharmacology
Plasmids
Polymorphism, Genetic
Pregnane X Receptor
Receptors, Steroid--genetics
Rifampin--pharmacology
Transcription Factors--metabolism
Transcriptional Activation
Two-Hybrid System Techniques