Both the suppressor of cytokine signaling 1 (SOCS-1) kinase inhibitory region and SOCS-1 mimetic bind to JAK2 autophosphorylation site: implications for the development of a SOCS-1 antagonist. [electronic resource]
- Journal of immunology (Baltimore, Md. : 1950) Apr 2007
- 5058-68 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
0022-1767
10.4049/jimmunol.178.8.5058 doi
Amino Acid Sequence Animals Cell Line Humans Interferon-Stimulated Gene Factor 3--metabolism Interferon-gamma--pharmacology Janus Kinase 2--metabolism Lymphocyte Activation--drug effects Macrophage Activation--drug effects Mice Mice, Inbred C57BL Molecular Sequence Data Peptide Fragments--pharmacology Phosphorylation Protein Kinase Inhibitors--metabolism STAT3 Transcription Factor--metabolism Suppressor of Cytokine Signaling 1 Protein Suppressor of Cytokine Signaling Proteins--antagonists & inhibitors src Homology Domains