Labrie, Philippe

In vitro activity of novel dual action MDR anthranilamide modulators with inhibitory activity on CYP-450 (Part 2). [electronic resource] - Bioorganic & medicinal chemistry Jun 2007 - 3854-68 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0968-0896

10.1016/j.bmc.2007.03.014 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--analysis
Biological Assay
Cell Line, Tumor
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--analysis
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Humans
Intestines--enzymology
Pyrazines--chemical synthesis
Quinolines--chemical synthesis
ortho-Aminobenzoates--chemistry