In vitro activity of novel dual action MDR anthranilamide modulators with inhibitory activity on CYP-450 (Part 2). [electronic resource]
- Bioorganic & medicinal chemistry Jun 2007
- 3854-68 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0968-0896
10.1016/j.bmc.2007.03.014 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--analysis Biological Assay Cell Line, Tumor Cytochrome P-450 CYP3A Cytochrome P-450 Enzyme Inhibitors Cytochrome P-450 Enzyme System--analysis Drug Resistance, Multiple--drug effects Drug Resistance, Neoplasm--drug effects Humans Intestines--enzymology Pyrazines--chemical synthesis Quinolines--chemical synthesis ortho-Aminobenzoates--chemistry