Wang, Gary T

Lead optimization of methionine aminopeptidase-2 (MetAP2) inhibitors containing sulfonamides of 5,6-disubstituted anthranilic acids. [electronic resource] - Bioorganic & medicinal chemistry letters May 2007 - 2817-22 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2007.02.062 doi


Aminopeptidases--antagonists & inhibitors
Lead--chemistry
Metalloendopeptidases--antagonists & inhibitors
Models, Molecular
Molecular Structure
Protein Conformation
Structure-Activity Relationship
Sulfonamides--chemistry
ortho-Aminobenzoates--chemistry