Parallel synthesis and SAR study of novel oxa-steroids as potent and selective progesterone receptor antagonists. [electronic resource]
- Bioorganic & medicinal chemistry letters May 2007
- 2531-4 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2007.02.013 doi
Animals Cell Line, Tumor Chemistry, Pharmaceutical--methods Complement C3--metabolism Drug Design Female Humans Mifepristone--pharmacology Models, Chemical Protein Binding Rats Receptors, Glucocorticoid--antagonists & inhibitors Receptors, Progesterone--antagonists & inhibitors Steroids--chemistry Structure-Activity Relationship