Battisti, Robert F

Modifying the sugar moieties of daunorubicin overcomes P-gp-mediated multidrug resistance. [electronic resource] - Molecular pharmaceutics - 140-53 p. digital

Publication Type: Journal Article

1543-8384

10.1021/mp060075v doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
ATP-Binding Cassette Transporters--chemistry
Bacterial Proteins--chemistry
Carbohydrate Metabolism
Cyclosporine--pharmacology
Cytotoxicity, Immunologic
Daunorubicin--analogs & derivatives
Disaccharides--metabolism
Drug Resistance, Multiple
Drug Resistance, Neoplasm
Gene Expression Regulation, Neoplastic
Humans
Inhibitory Concentration 50
K562 Cells
Monosaccharides--metabolism
Protein Structure, Secondary