Moerke, Nathan J

Small-molecule inhibition of the interaction between the translation initiation factors eIF4E and eIF4G. [electronic resource] - Cell Jan 2007 - 257-67 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

0092-8674

10.1016/j.cell.2006.11.046 doi


Animals
Antineoplastic Agents--chemistry
Cell Line, Transformed
Cell Line, Tumor
Cell Transformation, Neoplastic--drug effects
Drug Evaluation, Preclinical--methods
Eukaryotic Initiation Factor-4E--drug effects
Eukaryotic Initiation Factor-4G--drug effects
Feedback, Physiological--drug effects
Fluorescence Polarization Immunoassay--methods
Gene Expression Regulation, Neoplastic--drug effects
Humans
Hydrazones
Jurkat Cells
Mice
Models, Molecular
Nitro Compounds--chemistry
Oncogenes--drug effects
Peptide Fragments--genetics
Protein Binding--drug effects
Protein Biosynthesis--drug effects
RNA, Messenger--drug effects
Thiazoles--chemistry