Tang, Cuyue

Diclofenac hydroxylation in monkeys: efficiency, regioselectivity, and response to inhibitors. [electronic resource] - Biochemical pharmacology Mar 2007 - 880-90 p. digital

Publication Type: Journal Article

0006-2952

10.1016/j.bcp.2006.11.016 doi


Animals
Aryl Hydrocarbon Hydroxylases--antagonists & inhibitors
Catalysis
Chlorocebus aethiops
Cytochrome P-450 CYP2C9
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--physiology
Diclofenac--metabolism
Enzyme Inhibitors--pharmacology
Female
Humans
Hydroxylation
Kinetics
Macaca fascicularis
Macaca mulatta
Male
Microsomes, Liver--metabolism