TY - GEN AU - Gilbert,Adam M AU - Bursavich,Matthew G AU - Lombardi,Sabrina AU - Georgiadis,Katy E AU - Reifenberg,Erica AU - Flannery,Carl R AU - Morris,Elisabeth A TI - 5-((1H-pyrazol-4-yl)methylene)-2-thioxothiazolidin-4-one inhibitors of ADAMTS-5 SN - 0960-894X PY - 2007///0515 KW - ADAM Proteins KW - antagonists & inhibitors KW - ADAMTS4 Protein KW - ADAMTS5 Protein KW - Aggrecans KW - drug effects KW - Cartilage KW - Humans KW - Inhibitory Concentration 50 KW - Osteoporosis KW - drug therapy KW - Procollagen N-Endopeptidase KW - Structure-Activity Relationship KW - Thiazolidinediones KW - chemical synthesis N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2006.12.020 ER -