Structure-activity relationships of 3-aminoquinazolinediones, a new class of bacterial type-2 topoisomerase (DNA gyrase and topo IV) inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters Mar 2007
- 1312-20 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2006.12.005 doi
Amines--chemistry Anti-Bacterial Agents--chemical synthesis DNA Gyrase Gram-Positive Bacteria--drug effects Inhibitory Concentration 50 Quinazolinones--chemical synthesis Structure-Activity Relationship Topoisomerase II Inhibitors