Egbertson, Melissa S
A potent and orally active HIV-1 integrase inhibitor. [electronic resource]
- Bioorganic & medicinal chemistry letters Mar 2007
- 1392-8 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2006.11.080 doi
Administration, Oral
Animals
Cells, Cultured
HIV Integrase--drug effects
HIV Integrase Inhibitors--chemical synthesis
Humans
Inhibitory Concentration 50
Mutation
Naphthyridines--chemical synthesis
Rats
Structure-Activity Relationship