Egbertson, Melissa S

A potent and orally active HIV-1 integrase inhibitor. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2007 - 1392-8 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2006.11.080 doi


Administration, Oral
Animals
Cells, Cultured
HIV Integrase--drug effects
HIV Integrase Inhibitors--chemical synthesis
Humans
Inhibitory Concentration 50
Mutation
Naphthyridines--chemical synthesis
Rats
Structure-Activity Relationship