Sullivan, Susan K Allosteric and orthosteric binding modes of two nonpeptide human gonadotropin-releasing hormone receptor antagonists. [electronic resource] - Biochemistry Dec 2006 - 15327-37 p. digital Publication Type: Journal Article ISSN: 1520-4995 Standard No.: 10.1021/bi0617097 doi Subjects--Topical Terms: Allosteric Regulation--geneticsAnimalsBinding Sites--geneticsBinding, Competitive--geneticsCOS CellsCell Line, TumorChlorocebus aethiopsFurans--metabolismHormone Antagonists--metabolismHumansInhibitory Concentration 50Mutagenesis, Site-DirectedRadioligand AssayRatsReceptors, LHRH--agonistsStereoisomerismThymine--analogs & derivatives