Meyers, Kenneth M

Novel pyrazolopiperazinone- and pyrrolopiperazinone-based MCH-R1 antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2007 - 657-61 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2006.10.096 doi


Caco-2 Cells
Humans
Indicators and Reagents
Models, Molecular
Molecular Conformation
Piperazines--chemical synthesis
Pyrazoles--chemical synthesis
Pyrroles--chemical synthesis
Radioligand Assay
Receptor, Serotonin, 5-HT2C--drug effects
Receptors, Somatostatin--antagonists & inhibitors