Meyers, Kenneth M Novel pyrazolopiperazinone- and pyrrolopiperazinone-based MCH-R1 antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2007 - 657-61 p. digital Publication Type: Journal Article ISSN: 0960-894X Standard No.: 10.1016/j.bmcl.2006.10.096 doi Subjects--Topical Terms: Caco-2 CellsHumansIndicators and ReagentsModels, MolecularMolecular ConformationPiperazines--chemical synthesisPyrazoles--chemical synthesisPyrroles--chemical synthesisRadioligand AssayReceptor, Serotonin, 5-HT2C--drug effectsReceptors, Somatostatin--antagonists & inhibitors