Tian, Gaochao

Neurokinin-3 receptor-specific antagonists talnetant and osanetant show distinct mode of action in cellular Ca2+ mobilization but display similar binding kinetics and identical mechanism of binding in ligand cross-competition. [electronic resource] - Molecular pharmacology Mar 2007 - 902-11 p. digital

Publication Type: Journal Article

0026-895X

10.1124/mol.106.029868 doi


Animals
Binding, Competitive
CHO Cells
Calcium--metabolism
Cricetinae
Cricetulus
Kinetics
Neurokinin B--analogs & derivatives
Piperidines--metabolism
Quinolines--metabolism
Receptors, Neurokinin-3--antagonists & inhibitors