Tavares, Francis X

Potent, selective, and orally efficacious antagonists of melanin-concentrating hormone receptor 1. [electronic resource] - Journal of medicinal chemistry Nov 2006 - 7095-107 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm060572f doi


Administration, Oral
Animals
Anti-Obesity Agents--chemical synthesis
Biological Availability
CHO Cells
Cricetinae
Cricetulus
ERG1 Potassium Channel
Ether-A-Go-Go Potassium Channels--drug effects
Genes, Reporter
Half-Life
Humans
Mice
Mice, Obese
Models, Molecular
Pyrimidines--chemical synthesis
Rats
Receptors, Somatostatin--antagonists & inhibitors
Structure-Activity Relationship
Thiophenes--chemical synthesis