Tavares, Francis X Potent, selective, and orally efficacious antagonists of melanin-concentrating hormone receptor 1. [electronic resource] - Journal of medicinal chemistry Nov 2006 - 7095-107 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm060572f doi Subjects--Topical Terms: Administration, OralAnimalsAnti-Obesity Agents--chemical synthesisBiological AvailabilityCHO CellsCricetinaeCricetulusERG1 Potassium ChannelEther-A-Go-Go Potassium Channels--drug effectsGenes, ReporterHalf-LifeHumansMiceMice, ObeseModels, MolecularPyrimidines--chemical synthesisRatsReceptors, Somatostatin--antagonists & inhibitorsStructure-Activity RelationshipThiophenes--chemical synthesis