An opioid agonist that does not induce mu-opioid receptor--arrestin interactions or receptor internalization. [electronic resource]
- Molecular pharmacology Feb 2007
- 549-57 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
0026-895X
10.1124/mol.106.028258 doi
Analgesics, Opioid--pharmacology Animals Arrestin--drug effects Cell Line Diterpenes--pharmacology Diterpenes, Clerodane Drug Tolerance Endocytosis Humans Mice Morphine--pharmacology Protein Transport--drug effects Receptors, Opioid, mu--agonists Transfection