Frapolli, R

Pharmacokinetics and metabolism in mice of IDN 5390 (13-(N-Boc-3-i-butylisoserinoyl)-C-7,8-seco-10-deacetylbaccatin III), a new oral c-seco-taxane derivative with antiangiogenic property effective on paclitaxel-resistant tumors. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Dec 2006 - 2028-35 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0090-9556

10.1124/dmd.106.012153 doi


Angiogenesis Inhibitors--pharmacokinetics
Animals
Antineoplastic Agents, Phytogenic
Biological Availability
Bridged-Ring Compounds--pharmacokinetics
Cell Line, Tumor
Cell Proliferation--drug effects
Drug Resistance, Neoplasm
Feces--chemistry
Female
Mice
Mice, Inbred Strains
Microsomes, Liver--metabolism
Paclitaxel
Taxoids--pharmacokinetics
Tissue Distribution