High-content screening analysis of the p38 pathway: profiling of structurally related p38alpha kinase inhibitors using cell-based assays. [electronic resource]
- Assay and drug development technologies Aug 2006
- 397-409 p. digital
Publication Type: Journal Article
1540-658X
10.1089/adt.2006.4.397 doi
Animals Anisomycin--pharmacology Cell Line Cell Line, Tumor Chondrocytes--drug effects Dose-Response Relationship, Drug Drug Design Green Fluorescent Proteins--chemistry HSP27 Heat-Shock Proteins Heat-Shock Proteins--metabolism Humans Image Processing, Computer-Assisted--methods Interleukin-1beta--chemistry Intracellular Signaling Peptides and Proteins Lipopolysaccharides--pharmacology Mitogen-Activated Protein Kinase 14--antagonists & inhibitors Molecular Chaperones Molecular Structure Neoplasm Proteins--metabolism Phosphorylation--drug effects Protein Kinase Inhibitors--chemistry Protein Kinases--metabolism Protein Serine-Threonine Kinases Pyrimidinones--chemistry Signal Transduction--drug effects Structure-Activity Relationship Tumor Necrosis Factor-alpha--metabolism