Wood, Martyn D Aripiprazole and its human metabolite are partial agonists at the human dopamine D2 receptor, but the rodent metabolite displays antagonist properties. [electronic resource] - European journal of pharmacology Sep 2006 - 88-94 p. digital Publication Type: Comparative Study; Journal Article ISSN: 0014-2999 Standard No.: 10.1016/j.ejphar.2006.07.008 doi Subjects--Topical Terms: AmphetamineAnimalsAntipsychotic Agents--metabolismAripiprazoleBehavior, Animal--drug effectsBinding, CompetitiveBiotransformationCHO CellsCatalepsy--chemically inducedCricetinaeCricetulusDopamine D2 Receptor AntagonistsDyskinesia, Drug-Induced--etiologyGuanosine 5'-O-(3-Thiotriphosphate)--metabolismHeLa CellsHumansMaleMotor Activity--drug effectsOxidopaminePiperazines--metabolismQuinolones--metabolismRadioligand AssayRatsRats, Sprague-DawleyReceptors, Dopamine D2--agonistsSpecies SpecificityTransfection