D'Antona, Aaron M

A cannabinoid receptor 1 mutation proximal to the DRY motif results in constitutive activity and reveals intramolecular interactions involved in receptor activation. [electronic resource] - Brain research Sep 2006 - 1-11 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

0006-8993

10.1016/j.brainres.2006.05.042 doi


Amino Acid Motifs--drug effects
Amino Acid Sequence--physiology
Amino Acids--chemistry
Binding, Competitive--drug effects
Cannabinoids--metabolism
Cell Line
Cyclic AMP--metabolism
Cyclohexanes--pharmacology
Cyclohexanols
Guanosine 5'-O-(3-Thiotriphosphate)--pharmacology
Humans
Ligands
Molecular Structure
Mutation--genetics
Phenols--pharmacology
Piperidines--pharmacology
Pyrazoles--pharmacology
Radioligand Assay
Receptor, Cannabinoid, CB1--chemistry
Rimonabant