Levoye, Angélique The orphan GPR50 receptor specifically inhibits MT1 melatonin receptor function through heterodimerization. [electronic resource] - The EMBO journal Jul 2006 - 3012-23 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 0261-4189 Standard No.: 10.1038/sj.emboj.7601193 doi Subjects--Topical Terms: Arrestins--metabolismCell LineDimerizationDown-RegulationHumansLigandsMelatonin--metabolismMutationNerve Tissue Proteins--biosynthesisProtein BindingReceptor, Melatonin, MT1--antagonists & inhibitorsReceptor, Melatonin, MT2--antagonists & inhibitorsReceptors, G-Protein-Coupled--biosynthesisRecombinant Fusion Proteins--geneticsSignal Transductionbeta-Arrestins