Levoye, Angélique

The orphan GPR50 receptor specifically inhibits MT1 melatonin receptor function through heterodimerization. [electronic resource] - The EMBO journal Jul 2006 - 3012-23 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0261-4189

10.1038/sj.emboj.7601193 doi


Arrestins--metabolism
Cell Line
Dimerization
Down-Regulation
Humans
Ligands
Melatonin--metabolism
Mutation
Nerve Tissue Proteins--biosynthesis
Protein Binding
Receptor, Melatonin, MT1--antagonists & inhibitors
Receptor, Melatonin, MT2--antagonists & inhibitors
Receptors, G-Protein-Coupled--biosynthesis
Recombinant Fusion Proteins--genetics
Signal Transduction
beta-Arrestins