Mita, Sachiko

Inhibition of bile acid transport across Na+/taurocholate cotransporting polypeptide (SLC10A1) and bile salt export pump (ABCB 11)-coexpressing LLC-PK1 cells by cholestasis-inducing drugs. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Sep 2006 - 1575-81 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

0090-9556

10.1124/dmd.105.008748 doi


ATP Binding Cassette Transporter, Subfamily B, Member 11
ATP-Binding Cassette Transporters--antagonists & inhibitors
Animals
Bile Acids and Salts--metabolism
Biological Transport--drug effects
Cholestasis--etiology
Cyclosporine--toxicity
Dose-Response Relationship, Drug
Drug Evaluation, Preclinical--methods
Fluoresceins--metabolism
Kinetics
LLC-PK1 Cells
Organic Anion Transporters, Sodium-Dependent--antagonists & inhibitors
Oxadiazoles--metabolism
Rifampin--toxicity
Rifamycins--toxicity
Swine
Symporters--antagonists & inhibitors
Taurocholic Acid--analogs & derivatives
Transfection