Inhibition of bile acid transport across Na+/taurocholate cotransporting polypeptide (SLC10A1) and bile salt export pump (ABCB 11)-coexpressing LLC-PK1 cells by cholestasis-inducing drugs. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals Sep 2006
- 1575-81 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
0090-9556
10.1124/dmd.105.008748 doi
ATP Binding Cassette Transporter, Subfamily B, Member 11 ATP-Binding Cassette Transporters--antagonists & inhibitors Animals Bile Acids and Salts--metabolism Biological Transport--drug effects Cholestasis--etiology Cyclosporine--toxicity Dose-Response Relationship, Drug Drug Evaluation, Preclinical--methods Fluoresceins--metabolism Kinetics LLC-PK1 Cells Organic Anion Transporters, Sodium-Dependent--antagonists & inhibitors Oxadiazoles--metabolism Rifampin--toxicity Rifamycins--toxicity Swine Symporters--antagonists & inhibitors Taurocholic Acid--analogs & derivatives Transfection