Tauchi, Tetsuzo

The second generation of BCR-ABL tyrosine kinase inhibitors. [electronic resource] - International journal of hematology May 2006 - 294-300 p. digital

Publication Type: Journal Article; Review

0925-5710

10.1532/IJH97.06025 doi


Allosteric Regulation--drug effects
Antineoplastic Agents--chemistry
Binding Sites--drug effects
Drug Design
Drug Resistance, Neoplasm--drug effects
Fusion Proteins, bcr-abl
Gene Amplification--drug effects
Gene Expression Regulation, Leukemic--drug effects
Humans
Leukemia, Myelogenous, Chronic, BCR-ABL Positive--drug therapy
Mutation
Philadelphia Chromosome
Protein Binding--drug effects
Protein Kinase Inhibitors--chemistry
Protein Structure, Tertiary--drug effects
Protein-Tyrosine Kinases--antagonists & inhibitors