Tauchi, Tetsuzo
The second generation of BCR-ABL tyrosine kinase inhibitors. [electronic resource]
- International journal of hematology May 2006
- 294-300 p. digital
Publication Type: Journal Article; Review
0925-5710
10.1532/IJH97.06025 doi
Allosteric Regulation--drug effects
Antineoplastic Agents--chemistry
Binding Sites--drug effects
Drug Design
Drug Resistance, Neoplasm--drug effects
Fusion Proteins, bcr-abl
Gene Amplification--drug effects
Gene Expression Regulation, Leukemic--drug effects
Humans
Leukemia, Myelogenous, Chronic, BCR-ABL Positive--drug therapy
Mutation
Philadelphia Chromosome
Protein Binding--drug effects
Protein Kinase Inhibitors--chemistry
Protein Structure, Tertiary--drug effects
Protein-Tyrosine Kinases--antagonists & inhibitors