Yang, Lihu
Discovery of 3,5-bis(trifluoromethyl)benzyl L-arylglycinamide based potent CCR2 antagonists. [electronic resource]
- Bioorganic & medicinal chemistry letters Jul 2006
- 3735-9 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2006.04.045 doi
Animals
Binding Sites
CHO Cells--drug effects
Calcium--metabolism
Chemokine CCL2--antagonists & inhibitors
Cricetinae
Glycine--analogs & derivatives
Humans
Inhibitory Concentration 50
Models, Biological
Monocytes--drug effects
Receptors, CCR2
Receptors, Chemokine--antagonists & inhibitors