Yang, Lihu

Discovery of 3,5-bis(trifluoromethyl)benzyl L-arylglycinamide based potent CCR2 antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Jul 2006 - 3735-9 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2006.04.045 doi


Animals
Binding Sites
CHO Cells--drug effects
Calcium--metabolism
Chemokine CCL2--antagonists & inhibitors
Cricetinae
Glycine--analogs & derivatives
Humans
Inhibitory Concentration 50
Models, Biological
Monocytes--drug effects
Receptors, CCR2
Receptors, Chemokine--antagonists & inhibitors