TY  - GEN
AU  - Schwarz,Jacob B
AU  - Colbry,Norman L
AU  - Zhu,Zhijian
AU  - Nichelson,Brian
AU  - Barta,Nancy S
AU  - Lin,Kristin
AU  - Hudack,Raymond A
AU  - Gibbons,Sian E
AU  - Galatsis,Paul
AU  - DeOrazio,Russell J
AU  - Manning,David D
AU  - Vartanian,Mark G
AU  - Kinsora,Jack J
AU  - Lotarski,Susan M
AU  - Li,Zheng
AU  - Dickerson,Melvin R
AU  - El-Kattan,Ayman
AU  - Thorpe,Andrew J
AU  - Donevan,Sean D
AU  - Taylor,Charles P
AU  - Wustrow,David J
TI  - Carboxylate bioisosteres of pregabalin
SN  - 0960-894X
PY  - 2006///0802
KW  - Amines
KW  - chemical synthesis
KW  - Animals
KW  - Anticonvulsants
KW  - Binding Sites
KW  - Carboxylic Acids
KW  - chemistry
KW  - Cyclohexanecarboxylic Acids
KW  - Disease Models, Animal
KW  - Drug Evaluation, Preclinical
KW  - Epilepsy, Reflex
KW  - prevention & control
KW  - Gabapentin
KW  - Mice
KW  - Mice, Inbred DBA
KW  - Molecular Structure
KW  - Pregabalin
KW  - Protein Subunits
KW  - drug effects
KW  - Stereoisomerism
KW  - Structure-Activity Relationship
KW  - gamma-Aminobutyric Acid
KW  - analogs & derivatives
N1  - Publication Type: Journal Article
UR  - https://doi.org/10.1016/j.bmcl.2006.03.083
ER  -