Synthesis and evaluation of succinoyl-caprolactam gamma-secretase inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters May 2006
- 2357-63 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2006.01.055 doi
Alzheimer Disease--drug therapy Amyloid Precursor Protein Secretases Animals Aspartic Acid Endopeptidases Caprolactam--analogs & derivatives Cell Line Dogs Drug Design Drug Evaluation, Preclinical Endopeptidases--chemistry Enzyme Inhibitors--chemical synthesis Humans Molecular Conformation Stereoisomerism Structure-Activity Relationship Succinates--chemistry