Effect of P-glycoprotein on intestinal absorption and brain penetration of antiallergic agent bepotastine besilate. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals May 2006
- 793-9 p. digital
Publication Type: Journal Article
0090-9556
10.1124/dmd.105.007559 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism Adenosine Triphosphatases--metabolism Animals Anti-Allergic Agents--pharmacokinetics Autoradiography Biological Transport, Active Brain--metabolism Chromatography, Liquid Intestinal Absorption--drug effects Kinetics LLC-PK1 Cells Male Mass Spectrometry Mice Mice, Knockout Piperidines--pharmacokinetics Pyridines--pharmacokinetics Rats Rats, Sprague-Dawley Stimulation, Chemical Swine Terfenadine--analogs & derivatives Verapamil--pharmacology