Kajosaari, Lauri I
Pioglitazone, an in vitro inhibitor of CYP2C8 and CYP3A4, does not increase the plasma concentrations of the CYP2C8 and CYP3A4 substrate repaglinide. [electronic resource]
- European journal of clinical pharmacology Mar 2006
- 217-23 p. digital
Publication Type: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
ISSN: 0031-6970
Standard No.: 10.1007/s00228-005-0093-8 doi
Subjects--Topical Terms: Administration, Oral Adult Area Under Curve Aryl Hydrocarbon Hydroxylases--antagonists & inhibitors Blood Glucose--metabolism Capsules Carbamates--blood Chromatography, Liquid--methods Cross-Over Studies Cytochrome P-450 CYP2C8 Cytochrome P-450 CYP3A Cytochrome P-450 Enzyme Inhibitors Cytochrome P-450 Enzyme System--metabolism Drug Administration Schedule Enzyme Inhibitors--blood Female Gas Chromatography-Mass Spectrometry--methods Half-Life Humans Hypoglycemic Agents--administration & dosage In Vitro Techniques Male Pioglitazone Piperidines--blood Substrate Specificity Thiazolidinediones--administration & dosage