TY - GEN AU - Smith,Leon AU - Piatnitski,Evgueni L AU - Kiselyov,Alexander S AU - Ouyang,Xiaohu AU - Chen,Xiaoling AU - Burdzovic-Wizemann,Sabina AU - Xu,Yongjiang AU - Pan,Weitao AU - Chen,Xin AU - Wang,Ying AU - Rosler,Robin L AU - Patel,Sheetal N AU - Chiang,Hui-Hsien AU - Milligan,Daniel L AU - Columbus,John AU - Wong,Wai C AU - Doody,Jacqueline F AU - Hadari,Yaron R TI - Tricyclic azepine derivatives: pyrimido[4,5-b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors SN - 0960-894X PY - 2006///0417 KW - Adenosine Triphosphate KW - metabolism KW - Azepines KW - chemical synthesis KW - Binding Sites KW - Cell Proliferation KW - drug effects KW - Cells, Cultured KW - ErbB Receptors KW - antagonists & inhibitors KW - Humans KW - Molecular Structure KW - Phosphorylation KW - Protein Kinase Inhibitors KW - Protein Serine-Threonine Kinases KW - Protein-Tyrosine Kinases KW - Receptor, ErbB-2 KW - Structure-Activity Relationship KW - Substrate Specificity N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2005.12.018 ER -