Smith, Leon Tricyclic azepine derivatives: pyrimido[4,5-b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2006 - 1643-6 p. digital Publication Type: Journal Article ISSN: 0960-894X Standard No.: 10.1016/j.bmcl.2005.12.018 doi Subjects--Topical Terms: Adenosine Triphosphate--metabolismAzepines--chemical synthesisBinding SitesCell Proliferation--drug effectsCells, CulturedErbB Receptors--antagonists & inhibitorsHumansMolecular StructurePhosphorylation--drug effectsProtein Kinase Inhibitors--chemical synthesisProtein Serine-Threonine Kinases--antagonists & inhibitorsProtein-Tyrosine Kinases--antagonists & inhibitorsReceptor, ErbB-2--antagonists & inhibitorsStructure-Activity RelationshipSubstrate Specificity