Ngatcha, Béatrice Tchédam

3Beta-alkyl-androsterones as inhibitors of type 3 17beta-hydroxysteroid dehydrogenase: inhibitory potency in intact cells, selectivity towards isoforms 1, 2, 5 and 7, binding affinity for steroid receptors, and proliferative/antiproliferative activities on AR+ and ER+ cell lines. [electronic resource] - Molecular and cellular endocrinology Mar 2006 - 225-32 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0303-7207

10.1016/j.mce.2005.10.023 doi


17-Hydroxysteroid Dehydrogenases--antagonists & inhibitors
Androsterone--analogs & derivatives
Cell Proliferation--drug effects
Enzyme Inhibitors--chemical synthesis
Humans
Isoenzymes--antagonists & inhibitors
Receptors, Steroid--drug effects