Manetti, Fabrizio

Parallel solution-phase and microwave-assisted synthesis of new S-DABO derivatives endowed with subnanomolar anti-HIV-1 activity. [electronic resource] - Journal of medicinal chemistry Dec 2005 - 8000-8 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-2623

10.1021/jm050744t doi


Anti-HIV Agents--chemical synthesis
Cell Line
Drug Resistance, Multiple, Viral
HIV Reverse Transcriptase--metabolism
HIV-1--drug effects
Humans
Microwaves
Models, Molecular
Mutation
Pyrimidines--chemical synthesis
Pyrimidinones--chemical synthesis
Reverse Transcriptase Inhibitors--chemical synthesis
Solutions
Structure-Activity Relationship