Parallel solution-phase and microwave-assisted synthesis of new S-DABO derivatives endowed with subnanomolar anti-HIV-1 activity. [electronic resource]
- Journal of medicinal chemistry Dec 2005
- 8000-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0022-2623
10.1021/jm050744t doi
Anti-HIV Agents--chemical synthesis Cell Line Drug Resistance, Multiple, Viral HIV Reverse Transcriptase--metabolism HIV-1--drug effects Humans Microwaves Models, Molecular Mutation Pyrimidines--chemical synthesis Pyrimidinones--chemical synthesis Reverse Transcriptase Inhibitors--chemical synthesis Solutions Structure-Activity Relationship