In vitro and in vivo clinical pharmacology of dimethyl benzoylphenylurea, a novel oral tubulin-interactive agent. [electronic resource]
- Clinical cancer research : an official journal of the American Association for Cancer Research Dec 2005
- 8503-11 p. digital
Publication Type: Clinical Trial, Phase I; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1078-0432
10.1158/1078-0432.CCR-05-1037 doi
ATP Binding Cassette Transporter, Subfamily G, Member 2 ATP-Binding Cassette Transporters--metabolism Administration, Oral Animals Chromatography, High Pressure Liquid Cytochrome P-450 Enzyme System--metabolism Drug Therapy, Combination HIV Protease Inhibitors--pharmacology Humans In Vitro Techniques Mass Spectrometry Methylurea Compounds--blood Mice Microsomes, Liver--drug effects Neoplasm Proteins--metabolism Ritonavir--pharmacology Substrate Specificity Tubulin--metabolism