Rudek, Michelle A

In vitro and in vivo clinical pharmacology of dimethyl benzoylphenylurea, a novel oral tubulin-interactive agent. [electronic resource] - Clinical cancer research : an official journal of the American Association for Cancer Research Dec 2005 - 8503-11 p. digital

Publication Type: Clinical Trial, Phase I; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1078-0432

10.1158/1078-0432.CCR-05-1037 doi


ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--metabolism
Administration, Oral
Animals
Chromatography, High Pressure Liquid
Cytochrome P-450 Enzyme System--metabolism
Drug Therapy, Combination
HIV Protease Inhibitors--pharmacology
Humans
In Vitro Techniques
Mass Spectrometry
Methylurea Compounds--blood
Mice
Microsomes, Liver--drug effects
Neoplasm Proteins--metabolism
Ritonavir--pharmacology
Substrate Specificity
Tubulin--metabolism