Bleck, C

Essential role of the imidazoline moiety in the insulinotropic effect but not the KATP channel-blocking effect of imidazolines; a comparison of the effects of efaroxan and its imidazole analogue, KU14R. [electronic resource] - Diabetologia Dec 2005 - 2567-75 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

0012-186X

10.1007/s00125-005-0031-4 doi


Action Potentials--drug effects
Animals
Benzofurans--chemistry
Calcium--metabolism
Cell Line
Cytosol--metabolism
Imidazoles--chemistry
Imidazolines--chemistry
Insulin--metabolism
Insulin Secretion
Insulin-Secreting Cells--drug effects
Membrane Potentials--drug effects
Mice
Mice, Mutant Strains
Patch-Clamp Techniques
Potassium Channel Blockers--pharmacology
Potassium Channels--drug effects