Artemisinin and thiabendazole are potent inhibitors of cytochrome P450 1A2 (CYP1A2) activity in humans. [electronic resource]
- European journal of clinical pharmacology Nov 2005
- 755-61 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0031-6970
10.1007/s00228-005-0037-3 doi
Adult Antimalarials--pharmacology Antinematodal Agents--pharmacology Area Under Curve Artemisinins--pharmacology Caffeine--pharmacokinetics Chromatography, High Pressure Liquid Cytochrome P-450 CYP1A2--metabolism Cytochrome P-450 CYP1A2 Inhibitors Drug Interactions Enzyme Inhibitors--pharmacology Female Humans Male Mass Spectrometry Middle Aged Theophylline--metabolism Thiabendazole--metabolism