Synthesis and biological evaluation of 3-ethylidene-1,3-dihydro-indol-2-ones as novel checkpoint 1 inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters Jan 2006
- 421-6 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2005.09.064 doi
Cell Proliferation--drug effects Checkpoint Kinase 1 Crystallography, X-Ray Drug Design Drug Evaluation, Preclinical Enzyme Inhibitors--chemical synthesis HeLa Cells Humans Models, Molecular Molecular Structure Protein Kinases--drug effects Structure-Activity Relationship