Identification and initial evaluation of 4-N-aryl-[1,4]diazepane ureas as potent CXCR3 antagonists. [electronic resource]
- Bioorganic & medicinal chemistry letters Jan 2006
- 200-3 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2005.09.020 doi
Calcium--metabolism Cell Line Chemistry, Pharmaceutical--methods Chemokine CXCL11 Chemokines, CXC--chemistry Chemotaxis Dose-Response Relationship, Drug Drug Design Drug Evaluation, Preclinical Electrons Humans Inflammation Inhibitory Concentration 50 Models, Chemical Receptors, CXCR3 Receptors, Chemokine--antagonists & inhibitors Receptors, G-Protein-Coupled--metabolism Recombinant Proteins--chemistry Stereoisomerism T-Lymphocytes--cytology Urea--chemistry