Zhao, Chen

Synthesis and activity of N-acyl azacyclic urea HIV-1 protease inhibitors with high potency against multiple drug resistant viral strains. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2005 - 5499-503 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2005.08.093 doi


Aza Compounds--chemical synthesis
Drug Design
Drug Resistance, Multiple
HIV Protease Inhibitors--chemical synthesis
HIV-1--drug effects
Ligands
Microbial Sensitivity Tests
Models, Molecular
Ritonavir--chemical synthesis
Structure-Activity Relationship
Urea--analogs & derivatives