TY - GEN AU - Tehrani,Lida R AU - Smith,Nicholas D AU - Huang,Dehua AU - Poon,Steve F AU - Roppe,Jeffrey R AU - Seiders,Thomas Jon AU - Chapman,Deborah F AU - Chung,Janice AU - Cramer,Merryl AU - Cosford,Nicholas D P TI - 3-[Substituted]-5-(5-pyridin-2-yl-2H-tetrazol-2-yl)benzonitriles: identification of highly potent and selective metabotropic glutamate subtype 5 receptor antagonists SN - 0960-894X PY - 2005///1223 KW - Animals KW - Brain KW - drug effects KW - Excitatory Amino Acid Antagonists KW - chemical synthesis KW - Kinetics KW - Mice KW - Molecular Structure KW - Nitriles KW - chemistry KW - Pyridines KW - Rats KW - Receptor, Metabotropic Glutamate 5 KW - Receptors, Metabotropic Glutamate KW - antagonists & inhibitors KW - Sensitivity and Specificity KW - Structure-Activity Relationship KW - Substrate Specificity KW - Tetrazoles N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2005.07.062 ER -