3-O-acetyl-11-keto-boswellic acid decreases basal intracellular Ca2+ levels and inhibits agonist-induced Ca2+ mobilization and mitogen-activated protein kinase activation in human monocytic cells. [electronic resource]
- The Journal of pharmacology and experimental therapeutics Jan 2006
- 224-32 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0022-3565
10.1124/jpet.105.089466 doi
Anti-Inflammatory Agents Blotting, Western Calcium--metabolism Calcium Channel Agonists--pharmacology Cell Line Cell Membrane--drug effects Electrophoresis, Polyacrylamide Gel Enzyme Activation--drug effects Extracellular Signal-Regulated MAP Kinases--antagonists & inhibitors Humans In Vitro Techniques Inosine Triphosphate--metabolism Mitogen-Activated Protein Kinases--metabolism Monocytes--drug effects N-Formylmethionine Leucyl-Phenylalanine--pharmacology Neutrophils--drug effects Platelet Activating Factor--pharmacology Triterpenes--pharmacology p38 Mitogen-Activated Protein Kinases--antagonists & inhibitors